(r)-5-bromo-n-(1-ethyl-4-methylhexahydro-1h-1,4-diazepin-6-y...

Details (r)-5-bromo-n-(1-ethyl-4-methylhexahydro-1h-1,4-diazepin-6-y... (r)-5-bromo-n-(1-ethyl-4-methylhexahydro-1h-1,4-diazepin-6-y...

C - Chemistry, Metallurgy

07

D

C07D 401/12 (2006.01) A61K 31/55 (2006.01) C07D 243/08 (2006.01)

Patent

CA 2228056

The compound represented by formula (I) and physiologically acceptable acid- addition salts thereof. The compounds have an excellent antiemetic effect based on potent antagonism against serotonin S3 and dopamine D2 receptors and, therefore, are usable as an antiemetic agent in the treatment or prevention of various diseases and many digestive symptoms accompanying the administration of drugs, etc.

L'invention porte sur un composé de formule (1) et sur des sels d'addition d'acides pharmacocompatibles qui se caractérisent par leur excellent pouvoir antiémétique résultant de leur puissant antagonisme vis à vis des récepteurs de la sérotonine S¿3? et de la dopamine D¿2?. On peut les utiliser comme antiémétiques pour le traitement ou la prévention de différentes maladies et troubles digestifs liés à l'administration de médicaments.

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