C - Chemistry – Metallurgy – 07 – K
Patent
C - Chemistry, Metallurgy
07
K
C07K 5/062 (2006.01) A61K 31/381 (2006.01) A61K 31/5375 (2006.01) A61K 38/05 (2006.01) A61P 9/00 (2006.01) A61P 19/00 (2006.01) A61P 25/00 (2006.01) A61P 31/00 (2006.01) A61P 35/00 (2006.01) A61P 37/00 (2006.01) C07D 207/14 (2006.01) C07D 295/12 (2006.01) C07D 295/125 (2006.01) C07D 333/38 (2006.01) C07K 5/06 (2006.01) C07K 5/065 (2006.01) A61K 38/00 (2006.01)
Patent
CA 2380578
This invention relates to derivatives of alpha-amino acid amides, to pharmaceutical compositions containing such compounds, and to their use in medicine as inhibitors of cysteine proteases, particularly the cathepsins. A compound of formula (I) is described or a pharmaceutically acceptable salt, hydrate or solvate thereof. Pharmaceutically acceptable salts of the compounds of this invention include the sodium, potassium, magnesium, calcium, hydrogen chloride, tartaric acid, succinic acid, fumaric acid and p-toluenesulfonic acid salts.
La présente invention concerne des dérivés d'amides d'acide alpha aminés, des compositions pharmaceutiques contenant ces composés, et leur utilisation en médecine comme inhibiteurs des cystéine protéases, particulièrement les cathepsines. En outre, cette invention concerne un composé de la formule (I) ou un sel acceptable sur le plan pharmaceutique, un hydrate ou un solvate de celui-ci. Les sels acceptables sur le plan pharmaceutique de ces composés renferment du sodium, potassium, magnésium, calcium, chlorure d'hydrogène, acide tartrique, acide succinique, acide fumarique et des sels d'acides p-toluènesulfonique.
Ding Qizhu
Kaleta Jadwiga
Micetich Ronald George
Reddy Andhe V. N.
Singh Rajeshwar
Naeja Pharmaceutical Inc.
Riches Mckenzie & Herbert Llp
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