Selective inhibitors of neurotensin degrading enzymes

Details Selective inhibitors of neurotensin degrading enzymes Selective inhibitors of neurotensin degrading enzymes

C - Chemistry, Metallurgy

07

K

C07K 5/06 (2006.01) A61K 38/05 (2006.01) A61P 1/00 (2006.01) A61P 9/12 (2006.01) A61P 25/16 (2006.01) A61P 25/18 (2006.01) A61P 25/22 (2006.01) A61P 25/24 (2006.01) C07F 9/30 (2006.01) C07K 5/062 (2006.01) C07K 5/065 (2006.01) C07K 5/078 (2006.01)

Patent

CA 2670054

This invention concerns selective inhibitors of neurotensin degrading enzymes, to pharmaceutical compositions containing these compounds, to methods for preparing the compounds, methods for preparing novel intermediates useful for their synthesis, and methods for preparing compositions. The invention also relates to the uses of such compounds and compositions, particularly their use in the manufacture of medicaments for regulatingblood pressure orgastric emptying, or treating Parkinson s disease, anxiety, depression,orpsychosis. The compounds have the general formula (1) wherein the symbols have the meanings given in the specification.

L'invention concerne des inhibiteurs sélectifs d'enzymes dégradant la neurotensine, des compositions pharmaceutiques contenant ces composés, des procédés de préparation de ces composés, des procédés de préparation de nouveaux produits intermédiaires utiles dans la synthèse de ceux-ci et des procédés de préparation des compositions. L'invention concerne aussi l'utilisation de tels composés et compositions, en particulier leur utilisation dans la fabrication de médicaments destinés à réguler la pression artérielle ou le vidage gastrique, ou à traiter la maladie de Parkinson, l'anxiété, la dépression ou la psychose. Ces composés sont représentés par la formule générale (1), dans laquelle les symboles ont les notations indiquées dans la description.

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