C - Chemistry – Metallurgy – 07 – D
Patent
C - Chemistry, Metallurgy
07
D
C07D 405/06 (2006.01) A61K 31/4025 (2006.01) A61P 13/00 (2006.01)
Patent
CA 2480287
A stable solid hydrate of a muscarinic receptor antagonist in useful in the treatment of irritable bowel syndrome, diverticular disease, oesophageal achalasia, chronic obstructive airways disease, over active bladder (including symptoms of incontinence, urge and frequency), urinary incontinence, neurogenic urinary urgency or pollakiuria, treatment of bladder functional disorder, urinary leakage, painful or difficult urination caused by neurogenic bladder, spastic or hypertonic bladder, dysfunctional bladder syndrome, gastrointestinal disorders including gastrointestinal hyperactivity, and relaxing effect on intestinal smooth muscle cells.
Un hydrate solide stable d'antagoniste de récepteur muscarinique convient pour le traitement du syndrome du colon irritable, de la maladie diverticulaire, de l'achalasie oesophagienne, de la broncho-pneumopathie chronique obstructive, des troubles liés à la suractivité vésicale (comprenant les symptômes d'incontinence, de mictions impérieuses et fréquentes), de l'incontinence urinaire, de la miction impérieuse neurogène ou pollakiurie, le traitement des troubles fonctionnels de la vessie, des fuites urinaires, des douleurs ou des difficultés lors des mictions causées par une vessie neurogène, de la vessie spastique ou hypertonique, le syndrome de la vessie dysfonctionnelle, les troubles du tube digestif comprenant l'hyperactivité du tube digestif. Cet hydrate possède aussi un effet relaxant sur les cellules des muscles lisses.
Dunn Peter James
Matthews John George
Newbury Trevor Jack
O'connor Garry
Fetherstonhaugh & Co.
Novartis International Pharmaceutical Ltd.
LandOfFree
Stable hydrate of a muscarinic receptor antagonist does not yet have a rating. At this time, there are no reviews or comments for this patent.
If you have personal experience with Stable hydrate of a muscarinic receptor antagonist, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Stable hydrate of a muscarinic receptor antagonist will most certainly appreciate the feedback.
Profile ID: LFCA-PAI-O-1381293