Substituted 1-piperazinyl-triazolo-thieno-1,4- diazepines

Details Substituted 1-piperazinyl-triazolo-thieno-1,4- diazepines Substituted 1-piperazinyl-triazolo-thieno-1,4- diazepines

C - Chemistry, Metallurgy

07

D

260/239.3

C07D 495/14 (2006.01)

Patent

CA 1087182

ABSTRACT OF THE DISCLOSURE This invention relates to novel substituted 1-piperazino-4H-s-triazolo[3,4c]thieno[2,3e]1,4-diazepines of general formula Image (I) wherein R1 represents a hydrogen atom, an alkyl, halogenoalkyl,hydroxyalkyl or dialkylaminoalkyl group, a phenyl group optionally substituted by a methyl, methoxy or nitro group or by a halogen atom, or a pyridyl or pyrimidinyl group or a group of the formula R4- CO- (in which R4 represents a hydrogen atom, a C1 to C17 alkyl group, a C1 or C2 alkoxy group, or a phenyl, tolyl, methoxy- - 2 - phenyl, halogenophenyl, nitrophenyl or pyridyl group); R2 represents a hydrogen, fluorine, chlorine or bromine atom; and R3 represents a chlorine or bromine atom or an alkyl group] and, when R1 is hydrogen, alkyl, halogenoalkyl, hydroxyalkyl or dialkylaminoalkyl, acid addition salts thereof. The novel compounds exhibit pharmacological properties indicating their use as anxiolytics, tranquillizers, sedatives or neuroleptics. Processes for the preparation of the novel compounds and pharmaceutical compositions containing the novel compounds are described and claimed.

307798

Affiliated with

Also associated with

Rating

Substituted 1-piperazinyl-triazolo-thieno-1,4- diazepines does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Substituted 1-piperazinyl-triazolo-thieno-1,4- diazepines, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Substituted 1-piperazinyl-triazolo-thieno-1,4- diazepines will most certainly appreciate the feedback.

Rate now

Comments { 0 }

Profile ID: LFCA-PAI-O-533272