Substituted diketopiperazines as oxytocin antagonists

Details Substituted diketopiperazines as oxytocin antagonists Substituted diketopiperazines as oxytocin antagonists

C - Chemistry, Metallurgy

07

D

C07D 403/06 (2006.01) A61K 31/496 (2006.01) A61P 15/06 (2006.01)

Patent

CA 2571529

Compounds of formula (IA) wherein R1 is 2-indanyl, R2 is 1-methylpropyl, R3 is 1-methyl-indazol-5-yl, R4 represents methyl and R5 represents hydrogen or methyl, and pharmaceutically acceptable derivatives thereof are described, as are processes for their preparation, pharmaceutical compositions containing them and their use in medicine, particularly their use as oxytocin antagonists.

Cette invention concerne des composés représentés par la formule (IA), dans laquelle R1 représente 2-indanyle, R2 représente 1-méthylpropyle, R3 représente 1-méthyl-indazol-5-yle, R4 représente méthyle et R5 représente hydrogène ou méthyle, et des dérivés de ceux-ci acceptables sur le plan pharmaceutique, ainsi que des procédés pour leur préparation, des compositions pharmaceutiques les contenants et leur utilisation en médecine, notamment comme antagonistes des oxytocines.

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