C - Chemistry – Metallurgy – 07 – D
Patent
C - Chemistry, Metallurgy
07
D
C07D 215/04 (2006.01) A61K 31/47 (2006.01) A61P 33/02 (2006.01) C07D 215/02 (2006.01) C07D 215/12 (2006.01) C07D 215/14 (2006.01) C07D 215/24 (2006.01) C07D 405/06 (2006.01) C07F 7/08 (2006.01)
Patent
CA 2434063
The invention relates to the use of quinolines having general formula (I), wherein R¿1? denotes H; alkyl C¿1?-C¿15?; alkenyl or alkynyl C¿2?-C¿15?; -CHO; heteroaryl; alkyl C¿1?-C¿15? or alkenyl or alkynyl C¿2?-C¿7? comprising at least one substituent selected from among O, halogen, -OH, -CHO, -COOH, aryloxycarbonyl, alkyloxycarbonyl C¿2?-C¿8?, alkenyloxycarbonyl C¿3?-C¿9?, nitrile, aryl, heteroaryl, arylsulphone, alkylsulphone C¿1?-C¿7?, thioalkyl or aminoalkyl C¿1?-C¿7?; alkenyl C¿2?-C¿7? bearing at least one substituent selected from among NH¿2?, alcoxy C¿1?-C¿7?, phenoxy, cycloalkyl C¿3?-C¿6? or heteroaryloxy; alkenyl or alkynyl C¿2?-C¿15? comprising at least one trialkylsilyl C¿1?-C¿7?; R¿2?, in position 3, 6 or 8, denotes H; halogen; -OH; -CHO; -COOH; alkyl or alcoxy C¿1?-C¿7?; -NH2; alkenyl C¿2?-C¿7?; or alkynyl C¿2?-C¿10?; R¿1? and R¿2? do not both denote H. The invention is used for the preparation of a medicine to treat protozoan and retrovirus co-infections.
L'invention concerne l'utilisation de quinoléines de formule générale (I): dans laquelle R1 représente H; C1-C15; alkényle ou alkynyle C2-C15; -CHO; hétéroaryle; alkyle C1-C15 ou alkényle ou alkynyle C2-C7 portant au moins un substituant choisi parmi O, halogène, -OH, -CHO, -COOH, aryloxycarbonyle, alkyloxycarbonyle C2-C8, alkényloxycarbonyle C3-C9, nitrile, aryle, hétéroaryle, arylsulfone, alkylsulfone C1-C7, thioalkyle ou aminoalkyle C1-C7; alkényle C2-C7 portant au moins un substituant choisi parmi -NH2, alcoxy C1- C7, phénoxy, cycloalkyle C3-C6 ou hétéroaryloxy ; alkylène ou alkynyle C2-C15 portant au moins un trialkylsilyle C1-C7; R2, en position 3, 6 ou 8, représente H; halogène ; -OH; -CHO; -COOH; alkyle ou alcoxy C1-C7; -NH2 ; alkényle C2-C7; ou alkynyle C2-C10; R1 et R2 n'étant pas tous deux H; pour la préparation d'un médicament pour traiter les co-infections à protozoaires et à rétrovirus.
Fakhfakh Mohamed
Figadere Bruno
Fournet Alain
Franck Xavier
Hocquemiller Reynald
Centre National de La Recherche Scientifique
Institut de Recherche Pour Le Developpement (ird)
Macpherson Leslie & Tyerman Llp
LandOfFree
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