Thioquinolone derivatives

Details Thioquinolone derivatives Thioquinolone derivatives

C - Chemistry, Metallurgy

07

D

C07D 215/36 (2006.01) A61K 31/435 (2006.01) A61K 31/495 (2006.01) A61K 31/535 (2006.01) C07D 215/38 (2006.01) C07D 221/06 (2006.01) C07D 221/08 (2006.01) C07D 401/12 (2006.01) C07D 471/04 (2006.01) C07D 491/04 (2006.01) C07D 491/048 (2006.01)

Patent

CA 2201866

A thioquinolone derivative represented by general formula (I) and having a high selectivity and a potent antibacterial activity against Helicobacter pylori, wherein R1 and R2 represent each hydrogen or are combined together to represent -O-(CH2)2-; R3 represents halogen, C1-C12 alkyl, C1-C12 alkoxy, lower alkylsulfonyloxy, etc.; and R4 represents hydrogen or lower alkyl, or R4 and R3 are combined together to form a cyclohexene, benzene or pyridine ring.

On décrit un dérivé thioquinolone représenté par la formule générale (I), qui possède une sélectivité élevée ainsi qu'une puissante activité antibactérienne contre Helicobacter pylori. Dans cette formule, R¿1? et R¿2? représentent chacun hydrogène, ou bien combinés ensemble ils représentent -O-(CH¿2?)¿2?-; R¿3? représente halogène, alkyle C¿1?-C¿12?, alcoxy C¿1?-C¿12?, alkylsulfonyloxy inférieur, etc.; et R¿4? représente hydrogène ou alkyle inférieur, ou bien R¿4? et R¿3? sont combinés ensemble pour former un noyau cyclohexène, benzène ou pyridine.

Affiliated with

Also associated with

Rating

Thioquinolone derivatives does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Thioquinolone derivatives, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Thioquinolone derivatives will most certainly appreciate the feedback.

Rate now

Comments { 0 }

Profile ID: LFCA-PAI-O-2046818