Triazolylbenzophenone derivatives and production thereof

Details Triazolylbenzophenone derivatives and production thereof Triazolylbenzophenone derivatives and production thereof

C - Chemistry, Metallurgy

07

D

260/313.3, 260/2

C07D 403/00 (2006.01) C07D 239/86 (2006.01) C07D 239/92 (2006.01) C07D 249/08 (2006.01) C07D 249/16 (2006.01) C07D 265/30 (2006.01) C07D 295/00 (2006.01) C07D 401/00 (2006.01) C07D 405/00 (2006.01) C07D 409/00 (2006.01) C07K 5/06 (2006.01) C07K 5/065 (2006.01) A61K 38/00 (2006.01)

Patent

CA 1126274

TRIAZOLYLBENZOPHENONE DERIVATIVES AND PRODUCTION THEREOF Abstract: Triazolylbenzophenone derivatives of the formula: Image (wherein R represents hydrogen, C1-C6 alkyl, C1-C6 halo-alkyl, the group -(CH2)n-X-R5,or the group Image ; R5 represents hydrogen, C1-C6 alkyl, C2-C6 alkenyl, C2-C6 alkynyl, C6- C10 aryl, or C2-C8 acyl; X represents sulfur or oxygen; n represents 0, 1, 2, or 3; R6 and R7 each represents hydrogen or C1-C6alkyl: or the group R6-?-R7 represents pyrrolidino, piperidino, morpholino, or .gamma.-methylpiperazino; R1 represents hydrogen or halogen; R2 represents halogen, nitro, or trifluoromethyl; R3 represents C1-C6 alkyl, C1- C6 halo-alkyl, C1-C6 azido-alkyl, C6-C10 aryl, C2-C8 acyl or the group Image ; R4 and R8 each represents hydrogen, C1-C6 alkyl, or C7-C10 aralkyl; R9 represents hydrogen or C1-C6 alkyl; R10 represents hydrogen, C1-C6 alkyl, C7-C10 aralkyl, or C2-C11 .alpha.-amino-acyl; or the group R9-?-R10 represents phthalimido, pyrrolidino, piperidino, morpholino, or .gamma.-methylpiperazino) and their pharmaceutically acceptable acid addition salts, being useful as anxiolytics, sedatives, hypnotics, anti- convulsants, muscle relaxants, antidepressants,or their synthetic intermediates, are prepared. - 1 -

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