C - Chemistry – Metallurgy – 07 – D
Patent
C - Chemistry, Metallurgy
07
D
C07D 471/04 (2006.01) A61K 31/4375 (2006.01) A61K 31/496 (2006.01) A61K 31/7072 (2006.01) A61K 45/06 (2006.01) A61P 31/18 (2006.01) C07D 221/00 (2006.01)
Patent
CA 2418194
The present invention relates to tricyclic 2-pyridone compounds of formula (I): or stereoisomeric forms, stereoisomeric mixtures, or pharmaceutically acceptable salt forms thereof, which are useful as inhibitors of HIV reverse transcriptase, and to pharmaceutical compositions and diagnostic kits comprising the same, and methods of using the same for treating viral infection or as an assay standard or reagent.
L'invention concerne des composants pyridone-2 tricycliques de formule (I) : ou des formes stéréoisomériques, des mélanges stéréoisomériques ou des formes de sels pharmaceutiquement acceptables de ceux-ci, qui servent d'inhibiteurs de la transcriptase inverse HIV ou sont présents dans des préparations pharmaceutiques et des trousses de diagnostic. L'invention concerne également des procédés d'utilisation de ces composants afin de traiter une infection virale ou de servir de dosage biologique classique ou encore de réactif.
Arvanitis Argyrios
Cocuzza Anthony J.
Patel Mona
Rodgers James D.
Wang Haisheng
Bristol-Myers Squibb Pharma Company
Gowling Lafleur Henderson Llp
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