C - Chemistry – Metallurgy – 07 – D
Patent
C - Chemistry, Metallurgy
07
D
C07D 471/06 (2006.01) A61K 31/437 (2006.01) A61P 25/00 (2006.01) C07D 471/16 (2006.01)
Patent
CA 2716918
The present invention relates to compounds of formula (I) and pharmaceutically acceptable salts or tautomers thereof which are inhibitors of poly(ADP-ribose)polymerase (PARP) and thus useful for the treatment of cancer, inflammatory diseases, reperfusion injuries, ischaemic conditions, stroke, renal failure, cardiovascular diseases, vascular diseases other than cardiovascular diseases, diabetes mellitus, neurodegenerative diseases, retroviral infections, retinal damage, skin senescence and UV-induced skin damage, and as chemo-or radiosensitizers for cancer treatment.
La présente invention concerne des composés de formule (I) et des sels pharmaceutiquement acceptables ou tautomères de ceux-ci qui sont des inhibiteurs de poly(ADP-ribose)polymérase (PARP) et donc utiles pour le traitement du cancer, de maladies inflammatoires, de lésions de reperfusion, détats ischémiques, daccident cérébrovasculaire, dinsuffisance rénale, de maladies cardiovasculaires, de maladies vasculaires autres que des maladies cardiovasculaires, du diabète sucré, de maladies neurodégénératives, dinfections rétrovirales, de lésion rétinienne, du vieillissement de la peau et des lésions cutanées induites par les UV, et en tant que chimio- ou radiosensibilisateurs pour le traitement du cancer.
Bufi Laura Llauger
Ingenito Raffaele
Jones Philip
Ontoria Ontoria Jesus Maria
Scarpelli Rita
Istituto Di Ricerche Di Biologia Molecolare P. Angeletti Spa
Ogilvy Renault Llp/s.e.n.c.r.l.,s.r.l.
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