Substituted heterocycles and their use as chk1, pdk1 and pak...

Details Substituted heterocycles and their use as chk1, pdk1 and pak... Substituted heterocycles and their use as chk1, pdk1 and pak...

C - Chemistry, Metallurgy

07

D

C07D 495/04 (2006.01) A61K 31/404 (2006.01) A61K 31/4184 (2006.01) A61K 31/4355 (2006.01) A61K 31/4365 (2006.01) A61K 31/437 (2006.01) A61K 31/4439 (2006.01) C07D 209/08 (2006.01) C07D 209/10 (2006.01) C07D 209/12 (2006.01) C07D 209/14 (2006.01) C07D 235/18 (2006.01) C07D 401/04 (2006.01) C07D 491/04 (2006.01) C07D 513/04 (2006.01)

Patent

CA 2601983

This invention relates to novel compounds of Formula (I) and to their pharmaceutical compositions and to their methods of use. These novel compounds possess CHK1 kinase inhibitory activity, PDK1 inhibitory activity and Pak kinase inhibitory activity and are accordingly useful in the treatment and/or prophylaxis of cancer.

La présente invention concerne des nouveaux composés de formule (I) et leurs compositions pharmaceutiques ainsi que leurs procédés d~utilisation. Ces nouveaux composés possèdent une activité inhibant la CHK1 kinase, une activité inhibant la PDK1 et une activité inhibant la Pak kinase. Ils sont dès lors utiles dans le traitement et/ou la prophylaxie du cancer.

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