Salts of optically active sulfoxide derivative

Details Salts of optically active sulfoxide derivative Salts of optically active sulfoxide derivative

C - Chemistry, Metallurgy

07

D

C07D 495/10 (2006.01) A61K 31/5377 (2006.01)

Patent

CA 2290392

The below-described compound has good oral adsorption and exhibits markedly excellent antagonistic action against both NK1 receptors and NK2 receptors. Hydrochloride or fumarate of 1-{2-((2R)-(3,4-dichlorophenyl)-4-(3,4,5- trimethoxybenzoyl)morpholin-2-yl]ethyl}spiro[benzo(c)thiophene-1(3H),4'- piperidin]-(2S)-oxide.

Cette invention se rapporte à un hydrochlorure ou un fumarate de (2S)-oxyde de 1-{2-[(2R)- (3,4-dichlorophényl)-4- (3,4,5-triméthoxybenzoyl) morpholin-2-yl]éthyl} spiro[benzo(c)thiophène-1(3H),4'-pipéridine], ayant une bonne absorbabilité orale et de remarquables activités antagonistes sur les deux récepteurs NK1 et KN2.

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