Polycyclic compounds and processes for the preparation thereof

Details Polycyclic compounds and processes for the preparation thereof Polycyclic compounds and processes for the preparation thereof

C - Chemistry, Metallurgy

07

H

C07H 19/01 (2006.01) A61K 31/70 (2006.01) C07D 309/12 (2006.01) C07D 498/22 (2006.01) C07H 15/04 (2006.01)

Patent

CA 2122960

Polycyclic compounds and processes for the preparation thereof Abstract N-(tetrahydropyran-4-yloxy-alkanoyl)-staurosporin derivatives of formula I Image (I), wherein R1 is hydrogen, hydroxy, lower alkoxy or oxo, R2 is hydrogen or C1-4alkyl and R3 is hydrogen or C1-4alkyl, processes and novel intermediates for the preparation thereof and processes for the preparation of the intermediates are describe. The compounds of formula I inhibit the enzyme protein kinase C with a high degree of selectivity and can be used especially as tumour-inhibiting active ingredients.

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