Benzothiophenes with novel basic side chains

Details Benzothiophenes with novel basic side chains Benzothiophenes with novel basic side chains

C - Chemistry, Metallurgy

07

D

C07D 333/58 (2006.01) A61K 31/38 (2006.01) A61K 31/40 (2006.01) A61K 31/445 (2006.01) A61K 31/495 (2006.01) C07D 333/56 (2006.01) C07D 409/12 (2006.01) C07D 409/14 (2006.01)

Patent

CA 2215902

Compounds of formula (I), wherein R1 is selected from the group of H, OH, an alkoxy, OCOaryl, OCON(C1-C6alkyl)2, OCO(C1-C6alkyl), OCONH(C1-C6alkyl), OSO2(C1-C6alkyl), or halogen; R2 is selected from the group of H, OH, alkoxy, OCON(C1-C6alkyl)2, OCO(C1-C6alkyl), OCONH(C1-C6alkyl), OSO2(C4-C6alkyl), or halogen; with the proviso that when one of R1 and R2 is halogen, the other is not; and R3 is NR4R5, wherein R4 and R5 together with the nitrogen to which they are attached from a five- or six-membered heterocyclic ring as defined in the description.

La présente invention concerne des composés de la formule (I), dans laquelle R1 est choisi parmi: H, OH, un alcoxy, OCOaryle, OCON(alkyle C1-C6)2, OCO(alkyle C1-C6), OCONH(alkyle C1-C6), OSO2(alkyle C1-C6), ou un halogène; R2 est choisi parmi: H, OH, alcoxy, OCON(alkyle C1-C6)2, OCO(alkyle C1-C6), OCONH(alkyle C1-C6), OSO2(alkyle C4-C6), ou un halogène, à condition que R1 ou bien R2 soit halogène; et R3 est NR4R5, dans lequel R4 et R5 forment, avec l'azote auquel ils sont fixés, un noyau hétérocyclique à cinq ou six membres tel qu'il est défini dans la description.

Affiliated with

Also associated with

Rating

Benzothiophenes with novel basic side chains does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Benzothiophenes with novel basic side chains, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Benzothiophenes with novel basic side chains will most certainly appreciate the feedback.

Rate now

Comments { 0 }

Profile ID: LFCA-PAI-O-1484530