A - Human Necessities – 61 – K
Patent
A - Human Necessities
61
K
A61K 31/216 (2006.01) A61K 31/191 (2006.01) A61K 31/192 (2006.01) A61K 31/195 (2006.01) A61P 13/10 (2006.01)
Patent
CA 2524023
The present invention relates to a new field of indication for phenoxyacetic acid derivatives of the Formula I (see formula I) wherein X is a chiral carbon atom of R or S; Y is a chiral carbon atom of R or S; R1 is a hydroxy group, a C1-C6-alkoxy group, an aryl- C1-C6-alkoxy group, a primary amino group or a mono- or di (C1-C6-alkyl)amino group; one of the groups R2 and R3 is a hydrogen atom, the other group is a hydrogen atom , a halogen atom, a C1-C6-alkyl group, a trifluoromethyl group or a C1-C6- alkoxy group; and R4 is a halogen atom, a C1-C6-alkyl group, a halo (C1-C6-alkyl) group, a hydroxy group, a C1-C6-alkoxy group, an aryl- C1-C6-alkoxy group, a C1-C6-alkoxy group, a cyano group, a nitro group, an amino group, a mono- or di (C1-C6-alkyl)amino group, a carbamoyl group, a mono- or di (C1-C6-alkyl)carbamoyl group or the group - NHCOR5, where R5 is a hydrogen atom or a C1-C6-alkyl group; or a pharmaceutically acceptable salt thereof. It has now been found that the compounds described are suitable for the preparation of a medicament for treating hyperactive bladder (overactive bladder). Accordingly, by means of these active substances, a method is provided for treating this urological syndrome.
La présente invention se rapporte à un nouveau domaine d'indication pour des dérivés de l'acide phénoxyacétique comme décrit dans la demande de brevet européen EP 1095932. Il a été démontré que les composés décrit dans le brevet susmentionné se prêtent à la préparation d'un médicament traitant la vessie hyperactive. Dans cette même optique, au moyen de ces substances actives, on prévoit une méthode de traitement de ce syndrome urologique.
Kojima Masami
Yamazaki Yoshinobu
Kirby Eades Gale Baker
Kissei Pharmaceutical Co. Ltd.
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