1,3,5-trisubstituted 4,5-dihydro-1h-pyrazole derivatives...

Details 1,3,5-trisubstituted 4,5-dihydro-1h-pyrazole derivatives... 1,3,5-trisubstituted 4,5-dihydro-1h-pyrazole derivatives...

C - Chemistry, Metallurgy

07

D

C07D 231/06 (2006.01) A61K 31/415 (2006.01) A61K 31/454 (2006.01) A61P 25/00 (2006.01)

Patent

CA 2552940

The present invention relates to 1,3,5-trisubstituted 4,5-dihydro-1 H-pyrazole derivatives as CB1 antagonists, to methods for the preparation of these compounds and to novel intermediates useful for the synthesis of said pyrazole derivatives. The invention also relates to the use of a compound disclosed herein for the manufacture of a medicament giving a beneficial effect. The compounds have the general formula (I) wherein the symbols have the meanings given in the specification.

La présente invention concerne des dérivés de 4,5-dihydro-1h-pyrazole 1,3,5-trisubstitués présentant une activité antagonistique CB¿1?, des procédés de préparation de ces composés et de nouveaux intermédiaires utiles dans la synthèse de ces dérivés de pyrazole. L'invention concerne aussi l'utilisation d'un composé de l'invention, utile dans la fabrication d'un médicament qui présente un effet bénéfique. Les composés ont la formule générale (I) dans laquelle les symboles ont des significations déterminées dans la spécification.

Affiliated with

Also associated with

Rating

1,3,5-trisubstituted 4,5-dihydro-1h-pyrazole derivatives... does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with 1,3,5-trisubstituted 4,5-dihydro-1h-pyrazole derivatives..., we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and 1,3,5-trisubstituted 4,5-dihydro-1h-pyrazole derivatives... will most certainly appreciate the feedback.

Rate now

Comments { 0 }

Profile ID: LFCA-PAI-O-1821667