C - Chemistry – Metallurgy – 07 – D
Patent
C - Chemistry, Metallurgy
07
D
C07D 217/02 (2006.01) A61K 31/416 (2006.01) A61K 31/472 (2006.01) A61P 13/10 (2006.01) C07C 211/42 (2006.01) C07D 231/56 (2006.01) C07D 401/12 (2006.01) C07D 403/12 (2006.01)
Patent
CA 2526872
The present invention discloses novel compounds of general formula (I), or a pharmaceutically acceptable salt or prodrug thereof (in which X1 - X5, R5 - R8b, Z1 - Z2 and Ar1 are defined herein), a method for inhibiting the VR1 receptor in mammals using these compounds, a method for controlling pain in mammals, and pharmaceutical compositions including those compounds and a process for making those compounds.
L'invention concerne de nouveaux composés de la formule générale (I), ou d'un sel ou promédicament pharmaceutiquement acceptables de ceux-ci (X¿1? X¿5?, R¿5? R¿8b, Z1 Z2? et Ar¿1? étant tels que définis dans le descriptif), un procédé permettant d'inhiber le récepteur VR1 chez les mammifères au moyen de ces composés, un procédé permettant de maîtriser la douleur chez les mammifères, et des compositions pharmaceutiques comprenant ces composés ainsi qu'un processus de fabrication de ces composés.
Bayburt Erol K.
Chambournier Gilles
Cink Russell D.
Gomtsyan Arthur
Hsu Margaret
Abbott Laboratories
Torys Llp
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