Therapeutic agent for substance dependence

A - Human Necessities – 61 – K

Patent

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Details

A61K 31/343 (2006.01) A61P 25/30 (2006.01) A61P 25/32 (2006.01) A61P 25/36 (2006.01)

Patent

CA 2589289

[PROBLEMS] To provide a therapeutic agent for drug dependence which prevents the flash-back of or a relapse into a compulsive drug intake behavior based on the urge to, e.g., an addictive substance such as amphetamine, opium, barbiturate type morphine, psychedelic, cocaine, hemp, cannabins, alcohol, or volatile organic solvents. [MEANS FOR SOLVING PROBLEMS] (-)-1-(Benzofuran-2- yl)-2~propylaminopentane or a pharmacologically acceptable acid addition salt thereof is useful as a therapeutic agent for drug dependence which prevents the flash-back of or a relapse into a compulsive drug intake behavior based on the urge to, e.g., an addictive substance.

La présente invention a pour objet un agent thérapeutique pour le traitement de la dépendance à une drogue. Ledit agent empêche le phénomène de retour temporaire des effets (flash-back), ainsi que la rechute vers un comportement de prise compulsive de drogue. Il traite les dépendances à des substances telles que, par exemple, l'amphétamine, l'opium, les esters barbituriques de morphine, les drogues psychédéliques, la cocaïne, le chanvre, le cannabis, l'alcool, ou les solvants organiques volatils. Le (-)-1-(benzofuran-2-yl)-2-propylaminopentane, ou un sel d'addition acide de qualité pharmacologique dudit composé, peut ainsi être employé en tant qu'agent thérapeutique pour le traitement de la dépendance à une drogue, empêchant le phénomène de retour temporaire des effets (flash-back), ainsi que la rechute vers un comportement de prise compulsive de drogue, par le traitement de dépendances à diverses substances.

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