Substituted benzoylguanidines, process for their...

Details Substituted benzoylguanidines, process for their... Substituted benzoylguanidines, process for their...

C - Chemistry, Metallurgy

07

C

C07C 279/22 (2006.01) A01N 1/02 (2006.01) A61K 31/165 (2006.01) A61K 31/40 (2006.01) A61K 31/435 (2006.01) A61K 49/00 (2006.01) C07C 311/47 (2006.01) C07D 207/337 (2006.01) C07D 213/58 (2006.01) C07D 215/14 (2006.01) C07D 217/16 (2006.01)

Patent

CA 2163598

Substituted benzoylguanidines, process for their preparation, their use as a medicament or diagnostic, and medicament containing them Benzoylguanidines of the formula I Image I are described in which: R(1) is R(6)-CO or R(7)R(8)N-CO, and R(2) is defined as R(1) or is H, OH, Hal, CN, NO2, (perfluoro)alk(en)yl or -(CH)2R(15), or R(2) is (C1-C9) -heteroaryl, or R(2) is SR (18), -OR(18), -NR(18)R(19) or -CR(18)R(19)R(20); or R(2) is R(21)-SOm or R(22)R(23)N-SO2-, or R(2) is R(33)X-, where X is oxygen, S, NR(34), (D=O)A- or NR(34)C=MN(*)R(35)-, or R(2) is -SR(40), -OR(40), -NHR(40), -NR(40)R(41), -CHR(40)R(42), -CR(42)R(43)OH, -CCR(45), -CR(46)=CR(45) or -[CR(47)R(48)]u-CO- [CR(49)R(50)]v- R(44); or R(2) is R(55)-NH-SO2-, R(3), R(4) and R(5) are, independently of each other, defined as R(1) or R(2), where, however, at least one of the substituents R(2), R(3), R(4) and R(5) must be OH; as are the pharmaceutically tolerated salts thereof.

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