Use of pyrimidine derivatives for the treatment of egfr...

A - Human Necessities – 61 – K

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A61K 31/5377 (2006.01) A61P 35/00 (2006.01)

Patent

CA 2716518

The present invention relates to the use of compounds of formula (1), in the treatment of Epidermal Growth Factor Receptor (EGFR) family members dependent diseases or diseases that have acquired resistance to agents that target EGFR family members, use of said compounds for the manufacture of pharmaceutical compositions for the treatment of said diseases, combinations of said compounds with EGFR modulators for said use, methods of treating said diseases with said compounds and pharmaceutical preparations for the treatment of said diseases comprising said compounds alone or in combination, especially with an EGFR modulator.

La présente invention porte sur l'utilisation de composés de formule (I), dans le traitement de maladies dépendantes de membres de la famille des récepteurs de facteur de croissance épidermique (EGFR) ou de maladies qui ont acquis une résistance à des agents qui ciblent des membres de la famille EGFR, sur une utilisation desdits composés pour la fabrication de compositions pharmaceutiques pour le traitement desdites maladies, sur des combinaisons desdits composés avec des modulateurs d'EGFR pour ladite utilisation, sur des procédés de traitement desdites maladies avec lesdits composés et sur des préparations pharmaceutiques pour le traitement desdites maladies comprenant lesdits composés individuellement ou en combinaison, notamment avec un modulateur EGFR.

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