Diazepine derivatives

Details Diazepine derivatives Diazepine derivatives

C - Chemistry, Metallurgy

07

D

260/239.4

C07D 487/00 (2006.01) C07D 233/54 (2006.01) C07D 487/04 (2006.01) C07D 487/14 (2006.01) C07D 495/04 (2006.01) C07D 495/14 (2006.01) C07D 498/14 (2006.01) C07F 9/645 (2006.01) C07F 9/6561 (2006.01)

Patent

CA 1067491

ABSTRACT OF THE DISCLOSURE This invention is directed toward pharmacologically active com- pounds of the formula Image wherein A is Image ; R1 is selected from the group consisting of hydrogen, lower alkyl, phenyl, alkoxy lower alkyl, substituted phenyl, pyridyl and aral- kyl; R2 is selected from the group consisting of hydrogen and lower alkyl; R3 is selected from the group consisting of hydrogen and lower alkyl, R5 is selected from the group consisting of hydrogen, alkanoyloxy and hydroxy; R6 is selected from the group consisting of phenyl, mono-substituted phenyl, di- substituted phenyl, pyridyl, and mono-substituted pyridyl; and Image is selected from the group consisting of a) Image , b) Image , c) Image d) Image and wherein X is hydrogen, chlorine, bromine or iodine, T is hydrogen or lower alkyl and R4 is selected from the group consisting of hydrogen, halogen, nitro, cyano, trifluoromethyl, lower alkyl, substituted amino, amino, hydroxy lower alkyl and lower alkanoyl; and the pharmaceutically acceptable salts thereof, Also provided are methods for the preparation of these compounds as well as pharma- ceutical formulations which contain the active compounds of this invention. The compounds of the formulae illustrated above and their analogs are useful as anticonvulsants, muscle relaxants, anxiolytic and sedative agents.

235138

Affiliated with

Also associated with

Rating

Diazepine derivatives does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Diazepine derivatives, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Diazepine derivatives will most certainly appreciate the feedback.

Rate now

Comments { 0 }

Profile ID: LFCA-PAI-O-893990