3,3-disubstituted propylamines, their use and preparation

Details 3,3-disubstituted propylamines, their use and preparation 3,3-disubstituted propylamines, their use and preparation

C - Chemistry, Metallurgy

07

C

C07C 215/54 (2006.01) A61K 31/137 (2006.01) A61P 13/10 (2006.01) C07C 211/27 (2006.01) C07C 217/48 (2006.01) C07C 219/28 (2006.01) C07C 223/02 (2006.01)

Patent

CA 2284977

The invention relates to novel com-pounds of Formula (I) wherein R1, R2, R3, R4, R5, R6, R7 and Ar are as defined in claim 1, their salts with physiologically ac-ceptable acids and, when the compounds can be in the form of optical isomers, the racemic mixture and the individual enantiomers. The compounds have anticholinergic activity, and the invention also relates to the compounds of Formula (I) for use as therapeutically ac-tive substances, pharmaceutical compositions containing compounds of Formula (I), the use of the compounds of Formula (I) for preparing anticholinergic drugs, the use of the compounds of Formula (I) for treating urinary incontinence, and methods for preparing the compounds of Formula (I).

L'invention concerne de nouveaux composés de la formule (I) où R<1>, R<2>, R<3>, R<4>, R<5>, R<6>, R<7> et Ar sont tels que définis dans la 1ère revendication. L'invention concerne également leurs sels aux acides physiologiquement tolérables et, lorsque les composés peuvent être sous la forme d'isomères optiques, le mélange racémique et les énantiomères individuels. Ces composés ont une activité anticholinergique. En outre, l'invention concerne les composés de la formule (I), destinés à être utilisés comme substances à action thérapeutique, les compositions pharmaceutiques contenant des composés de la formule (I), l'utilisation des composés de la formule (I) dans la préparation de médicaments anticholinergiques, l'utilisation des composés de la formule (I) dans le traitement de l'incontinence urinaire et des procédés de préparation des composés de la formule (I).

Affiliated with

Also associated with

Rating

3,3-disubstituted propylamines, their use and preparation does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with 3,3-disubstituted propylamines, their use and preparation, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and 3,3-disubstituted propylamines, their use and preparation will most certainly appreciate the feedback.

Rate now

Comments { 0 }

Profile ID: LFCA-PAI-O-1658388