C - Chemistry – Metallurgy – 07 – D
Patent
C - Chemistry, Metallurgy
07
D
C07D 307/64 (2006.01) A01N 33/22 (2006.01) A01N 43/00 (2006.01) A01N 43/08 (2006.01) A01N 43/10 (2006.01) A01N 43/40 (2006.01) A01N 43/50 (2006.01) A01N 43/54 (2006.01) A01N 43/56 (2006.01) A01N 43/58 (2006.01) A01N 43/64 (2006.01) A01N 43/66 (2006.01) A01N 43/707 (2006.01) A01N 43/713 (2006.01) A01N 43/74 (2006.01) A01N 43/80 (2006.01) A01N 43/82 (2006.01) C07C 17/087 (2006.01) C07C 17/23 (2006.01) C07C 317/14 (2006.01) C07C 323/05 (2006.01) C07C 323/09 (2006.01) C07D 213/62 (2006.01) C07D 213/70 (2006.01)
Patent
CA 2182520
A compound of formula (I), or a salt thereof, whenein n is 0, 1 or 2; and R is a group of formulae (II) to (XXI), wherein: the S(O)nCH2CH2CH=CF2 group is at least one of R1 (when attached to a carbon atom), R2, R3, R4, R5 or R6; R1 (when attached to a carbon atom), R2, R3, R4, R5 and R6 are each independentiy hydrogen, optionally substituted alkyl, optionally substituted alkenyl, alkynyl, cycloalkyl, alkylcycloalkyl, alkoxy, alkenyloxy, alkynyloxy, hydroxyalkyl, alkoxyalkyl, optionally substituted aryl, optionally substituted arylalkyl, optionally substituted heteroaryl, optionally substituted heteroarylalkyl, optionally substituted aryloxy, optionaily substituted arylalkoxy, optionally substituted aryloxyalkyl, optionally substituted heteroaryloxy, optionally substituted heteroarylalkoxy, optionally substituted heteroaryloxyalkyl, haloalkyl, haloalkenyl, haloalkynyl, haloalkoxy, haloalkenyloxy, haloalkynyloxy, halogen, hydroxy, cyano, nitro, -NR7R8, -NR7COR8, -NR7CSR8, -NR7SO2R8, -N(SO2R7)(SO2R8), -COR7, -CONR7R8, -alkylCONR7R8, CR7NR8, -COOR7, -OCOR7, -SR7, -SOR7, SO2R7, -alkylSR7, -alkylSOR7, -alkylSO2R7, -OSO2R7, -SO2NR7R8, -CSNR7R8, SiR7R8R9, -OCH2CO2R7, -OCH2CH2CO2R7, -CONR7SO2R8, -alkylCONR7SO2R8, -NHCONR7R8, -NHCSNR7R8, or an adjacent pair of R1, R2 R3, R4, R5 and R6 when taken together form a fused 5- or 6-membered carbocyclic or heterocyclic ring; R1 (when attached to a nitrogen atom) is hydrogen, optionally substituted alkyl, cycloalkyl, alkylcycloalkyl, hydroxyalkyl, alkoxyalkyl, optionally substituted aryl, optionally substituted arylalkyl, optionally substituted aryloxyalkyl, optionally substituted heteroaryl, optionally substituted heteroarylakyl, optionally substituted heteroaryloxyalkyl, haloalkyl, hydroxy, cyano, nitro, -NR7R8, -NR7COR8, NR7CSR8, -NR7COOR8, -NR7SO2R8, -N(SO2R7)(SO2R8), -COR7, -CONR7R8, -alkylCONR7R8, -CR7NR8, -COOR7, -OCOR7, -SOR7 -SO2R7 -alkylSR7 -alkylSOR7 -alkylSO2R7, -OSO2R7, - SO2NR7NR8, -SR7, -SOR7, -SO2R7, -CSNR7R8, -SiR7R8R7, -OCH2CO2R7, -OCH2CH2CO2R7, CONR7SO2R8, -alkylCONR7SO2R8, -NHCOR7R8, or -NHCSR7R8; and R7, R8 and R9 are each independently hydrogen, optionally substituted alkyl, optionally substituted alkenyl, alkynyl, optionally substituted aryl or optionally substituted arylaikyl, haloalkyl, haloalkenyl, haloalkynyl, halogen, or hydroxy.
Dans un composé de formule (I) ou dans un de ses sels, n vaut 0, 1 ou 2; et R représente un groupe de formule (II) à (XXI), où le groupe S(O)nCH2CH2CH=CF2 correspond au moins à une des références R1 (lorsqu'il est lié à un atome de carbone), R2, R3, R4, R5 ou R6 lesquels représentent chacun indépendamment hydrogène, ou bien alkyle, ou alcényle éventuellement substitué, alkynyle, cycloalkyle, alkylcycloalkyle, alcoxy, alkényloxy, alkynyloxy, hydroxyalkyle, alcoxyalkyle, ou bien aryle, arylalkyle, hétéroaryle, hétéroarylalkyle, aryloxy, arylalcoxy, aryloxyalkyle, hétéroaryloxy, hétéroarylalcoxy ou hétéroaryloxyalkyle éventuellement substitué, ou bien haloalkyle, haloalkényle, haloalkynyle, haloalcoxy, haloalkényloxy, haloalkynyloxy, halogène, hydroxy, cyano, nitro, -NR7R8, -NR7COR8, -NR7CSR8, -NR7SO2R8, -N(SO2R7)(SO2R8), -COR7, -CONR7R8, -alkylCONR7R8, CR7NR8, -COOR7, -OCOR7, -SR7, -SOR7, SO2R7, -alkylSR7, -alkylSOR7, -alkylSO2R7, -OSO2R7, -SO2NR7R8, -CSNR7R8, SiR7R8R9, -OCH2CO2R7, -OCH2CH2CO2R7, -CONR7SO2R8, -alkylCONR7SO2R8, -NHCONR7R8, -NHCSNR7R8; ou bien une paire adjacente de R1, R2, R3, R4, R5 et R6, puis conjointement, forment un cycle carbocyclique ou hétérocyclique fusionné à 5 ou 6 membres. R1 (lorsqu'il est lié à un atome d'azote) représente hydrogène, alkyle éventuellement substitué, cycloalkyle, alkylcycloalkyle, hydroxyalkyle, alcoxyalkyle, ou bien aryle, arylalkyle, aryloxyalkyle, hétéroaryle, hétéroarylakyle ou hétéroaryloxyalkyle éventuellement substitués, haloalkyle, hydroxy, cyano, nitro, -NR7R8, -NR7COR8, NR7CSR8, -NR7COOR8, -NR7SO2R8, -N(SO2R7)(SO2R8), -COR7, -CONR7R8, -alkylCONR7R8, -CR7NR8, -COOR7, -OCOR7, -SOR7, -SO2R7, -alkylSR7, -alkylSOR7, -alkylSO2R7, -OSO2R7, -SO2NR7NR8, -SR7, -SOR7, -SO2R7, -CSNR7R8, -SiR7R8R7, -OCH2CO2R7, -OCH2CH2CO2R7, -CONR7SO2R8, -alkylCONR7SO2R8, -NHCOR7R8, ou -NHCSR7R8; et R7, R8 et R9 représentent chacun indépendamment hydrogène, ou bien alkyle ou alcényle éventuellement substitué, alkynyle, ou bien aryle ou arylalkyle éventuellement substitué, haloalkyle, haloalkényle, haloalkynyle, halogène, ou hydroxy.
Bansal Harjinder Singh
Dowling Alan John
Fitzjohn Steven
Godfrey Christopher Richard Ayles
Hotson Matthew Brian
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