Aminoquinoline derivatives and their use as adenosine a3...

Details Aminoquinoline derivatives and their use as adenosine a3... Aminoquinoline derivatives and their use as adenosine a3...

C - Chemistry, Metallurgy

07

D

C07D 215/48 (2006.01) A61K 31/4706 (2006.01) A61P 43/00 (2006.01) C07D 213/85 (2006.01) C07D 215/46 (2006.01) C07D 401/12 (2006.01) C07D 405/12 (2006.01) C07D 405/14 (2006.01) C07D 409/12 (2006.01) C07D 409/14 (2006.01)

Patent

CA 2448561

The invention provides compounds of general formula (I), (see formula I) wherein R4 and R5 form together an 1,3-butadienyl group, optionally substituted by a methylenedioxy group or one or more straight or branched C1-4 alkyl group, straight or branched C1-4 alkoxy group, hydroxy group or halogen atom. The compounds of the invention are strong adenosine A3 receptor ligands preferably antagonists.

Cette invention se rapporte à des composés représentés par la formule générale (I), où R<4> et R<5> représentent un atome d'hydrogène ou forment ensemble un groupe 1,3-butadiényle, éventuellement substitué par un groupe méthylène-dioxy ou l'un et/ou l'autre des radicaux suivants: groupe alkyle C1-C4 droit ou ramifié, groupe alcoxy C1-C4 droit ou ramifié, groupe hydroxy ou atome d'halogène. Ces composés constituent de puissants ligands, de préférence antagonistes, du récepteur d'adénosine A3.

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