Heteroaryl derivatives as superior ligands for nociceptin...

Details Heteroaryl derivatives as superior ligands for nociceptin... Heteroaryl derivatives as superior ligands for nociceptin...

C - Chemistry, Metallurgy

07

D

C07D 451/06 (2006.01) A61K 31/46 (2006.01) A61K 31/506 (2006.01)

Patent

CA 2465871

Novel compounds of the formula (I), wherein R is optionally substituted heteroaryl or (a); R1 is H or C1-C6 alkyl; and R2 and R3 are -CH3, -OCH3 or halo; or a pharmaceutically acceptable salt or solvate thereof, pharmaceutical compositions therefore, and the use of said compounds in the treatment of pain, anxiety, cough, asthma, depression and alcohol abuse are disclosed.

Nouveaux composés correspondant à la formule (I), dans laquelle R est un hétéroaryle éventuellement substitué ou (a); R<1> est H ou alkyle C1-C6; et R<2> et R<3> sont -CH3, -OCH3 ou halo; ou un sel pharmaceutiquement acceptable ou un solvate, et l'utilisation de ces composés dans le traitement de la douleur, de l'anxiété, de la toux, de l'asthme, de la dépression et de l'abus d'alcool.

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