Inhibitors of the enzymatic activity of psa

Details Inhibitors of the enzymatic activity of psa Inhibitors of the enzymatic activity of psa

C - Chemistry, Metallurgy

07

D

C07D 205/04 (2006.01) A61K 31/00 (2006.01) A61K 31/397 (2006.01) A61K 31/4035 (2006.01) A61K 31/422 (2006.01) A61K 31/43 (2006.01) A61K 31/4439 (2006.01) A61K 31/545 (2006.01) C07D 205/08 (2006.01) C07D 401/14 (2006.01) C07D 403/04 (2006.01) C07D 413/04 (2006.01) C07D 413/14 (2006.01)

Patent

CA 2274958

This invention is directed to novel azetidinone compounds, to certain intermediates and processes for preparing these azetidinone compounds, and to formulations containing the same. The present invention also relates to the use of these azetidinones as inhibitors of the enzymatic activity of Prostate- Specific Antigen (PSA) as well as for treating prostatic cancer (Pca), Pca metastasis, benign prostatic hyperplasia (BPH) and breast cancer (Bc). Another aspect of the invention relates to inventive methods for treating Pca, Pca metastasis, BPH and Bc by administering any PSA inhibiting compound.

La présente invention concerne des composés azétidinone, certains intermédiaires et procédés permettant d'élaborer de tels composés azétidinone, et des formulations contenant ces composés et intermédiaires. L'invention concerne également l'utilisation de ces azétidinones comme inhibiteurs de l'activité enzymatique de l'antigène PSA (Prostate-Specific Antigen) ainsi qu'un traitement contre le cancer de la prostate (Pca), contre les métastases Pca, contre l'hyperplasie prostatique bénigne (BPH) et contre le cancer du sein (Bc). Un autre aspect de l'invention concerne des procédés nouveaux permettant de traiter le cancer de la prostate (Pca), les métastases Pca, l'hyperplasie prostatique bénigne (BPH) et le cancer du sein (Bc) par administration de n'importe quel composé inhibiteur du PSA.

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