C - Chemistry – Metallurgy – 07 – D
Patent
C - Chemistry, Metallurgy
07
D
C07D 487/08 (2006.01) A61K 31/4995 (2006.01) A61K 31/55 (2006.01) A61K 49/00 (2006.01) A61P 25/04 (2006.01) C07D 487/18 (2006.01)
Patent
CA 2724086
Diazapolycyclic compounds having affinity for the opioidergic receptors, preferably for the delta opioidergic receptors, with central and/or peripheral activity, having formula: A1-D1-T1 (I) wherein: - A1 is a group of formula (II): (see formula II) wherein: R1 is phenyl wherein one of the ring hydrogen atoms is substituted with a group selected from C(O)R', C(O)OR', C(O)NHR' or C(O)NR3R4, R', R3 and R4, being as defined in the application; R2 is phenyl, optionally substituted - D1 is a diazapolycyclic group - T1 is a group selected from H, alkyl, alkenyl, alkynyl and from the following optionally substituted groups: cycloalkyl, heterocycloalkyl, aryl, heteroaryl, cycloalkylalkyl, heterocycloalkylalkyl, arylalkyl or heteroarylalkyl, and their hydrates and solvates and pharmaceutically acceptable salts.
Lazzari Paolo
Loriga Giovanni
Murineddu Gabriele
Pani Luca
Pinna Gerard Aime
Gowling Lafleur Henderson Llp
Neuroscienze Pharmaness S.c. A. R.l.
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