Polymer particle delivery compositions and methods of use

A - Human Necessities – 61 – K

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A61K 9/50 (2006.01)

Patent

CA 2596011

The present invention provides biodegradable polymer particle delivery compositions based on polymers, such as polyester amide (PEA) and polyester urethane (PEUR) polymers, that contain amino acids in the polymer. The polymer particle delivery compositions can be formulated as a liquid dispersion of polymer particles with the bioactive agents dispersed in the particle or conjugated attached to polymer molecules or particle surfaces. The bioactive agents can include drugs, polypeptides, DNA and cells for cell-based therapies using particles sized for local, mucosal or circulatory delivery. Methods of treating a disease by administering to a subject the polymer particle delivery composition, which incorporates a bioactive agent suitable for treatment of the disease, or its symptoms, are also included.

La présente invention concerne des compositions d'administration particulaires, polymériques, biodégradables, à base de polymères, tels que des polymères à base de polyester-amide (PEA) et de polyesteruréthane (PEUR), contenant des acides aminés dans le polymère. Ces compositions d'administration particulaires, polymériques, peuvent être préparées sous forme de dispersion liquide de particules polymériques, avec les agents bioactifs dispersés dans la particule ou conjugués et fixés à des molécules polymériques ou des surfaces particulaires. Les agents bioactifs utilisés peuvent être des médicaments, des polypeptides, de l'ADN et des cellules pour des thérapies à base de cellules dans lesquelles sont utilisées des particules dont les dimensions conviennent pour une administration locale, par la muqueuse ou par voie circulatoire. L'invention concerne également des méthodes destinées au traitement d'une maladie, consistant à administrer à un sujet la composition d'administration particulaire, polymérique, contenant un agent bioactif convenant au traitement de cette maladie ou de ses symptômes.

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