Prodrugs of er.beta-selective substances, process for their...

Details Prodrugs of er.beta-selective substances, process for their... Prodrugs of er.beta-selective substances, process for their...

C - Chemistry, Metallurgy

07

J

C07J 41/00 (2006.01) A61K 31/565 (2006.01) A61P 5/30 (2006.01)

Patent

CA 2630438

The invention relates to prodrugs of 8-.beta.-substituted estratrienes of general formula (I) in which the Z group is bonded to the steroid, method for production thereof, pharmaceutical compositions comprising said compounds and use thereof. Said compounds of general formula (I) do not bind to .alpha.- and/or .beta.- estrogen receptors, but to carboanhydrases and inhibit said enzymes.

L'invention concerne des promédicaments d'estratriènes à substitution 8ß de formule (I), dans lesquels le groupe Z est lié au stéroïde, (I). La présente invention porte également sur des procédés pour les réaliser, sur des compositions pharmaceutiques contenant ces composés et sur leur utilisation. Les composés de l'invention de formule (I) ne se lient pas au récepteur d'oestrogène alpha et/ou bêta, mais ils se lient à des carboanhydrases et inhibent ces enzymes.

Affiliated with

Also associated with

Rating

Prodrugs of er.beta-selective substances, process for their... does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Prodrugs of er.beta-selective substances, process for their..., we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Prodrugs of er.beta-selective substances, process for their... will most certainly appreciate the feedback.

Rate now

Comments { 0 }

Profile ID: LFCA-PAI-O-1652305